22- Regio- and chemoselective covalent immobilization of proteins through unnatural amino acids. Cécile Gauchet, Guillermo R. Labadie and C. Dale Poulter. J. Am. Chem. Soc. 128, 9274-5 (2006) doi: 10.1021/ja061131o
23- An efficient approach toward the synthesis of the A/B rings of Ouabain. María Fernanda Plano, Guillermo R. Labadie, Manuel Gonzalez Sierra and Raquel M. Cravero. Tetrahedron Lett. 47, 7447-7449 (2006) doi: 10.1016/j.tetlet.2006.08.047
24- A simple synthesis of a model of the tetracyclic bis-ketal lactone mainframe of saudin. Guillermo R. Labadie, Liliana E. Luna, Raquel M. Cravero, Manuel González-Sierra Helv. Chim. Acta 89, 2732-2737 (2006) doi: 10.1021/ja061131o
25- Design, synthesis and evaluation of omega-azido and alkynyl farnesyl diphosphate analogs as protein farnesyl transferase substrates. Guillermo R. Labadie, Rajesh Viswanathan and C. Dale Poulter. J. Org. Chem. 72, 9291- 9297 (2007) doi: 10.1021/jo7017747
26- Semisynthetic Studies on the Manzamine Alkaloids. Khalid A. El Sayed, Ashraf A. Khalil, Muhammad Yousaf, Guillermo Labadie, Gundluru M. Kumar, Scott G. Franzblau, Alejandro M. S. Mayer, Mitchell A. Avery, and Mark T. Hamann. J. Nat. Prod. 71, 300-308 (2008) doi: 10.1021/np0703702
27- Preparation of phenyl-butyraldehydes using a base-catalyzed aromatization of dienones. María Fernanda Plano, Guillermo R. Labadie, Raquel M. Cravero. Tetrahedron Lett. 49, 2872–2874 (2008) doi: 10.1016/j.tetlet.2008.03.038
28- Biosynthesis of TDP-L-megosamine: pathway elucidation and megalomicin A production in Escherichia coli. Mariana Useglio, Salvador Peirú, Eduardo Rodríguez, Guillermo R. Labadie, John R. Carney, and Hugo Gramajo Appl. Environ. Microbiol. 76, 3869-3077 (2010) doi: 10.1128/AEM.03083-09
29- Identificación, cuantificación y determinación de variabilidad en el tiempo de componentes insolubles de biodiesel de soja comerciales argentinos. Rodolfo Cabrera, Pablo Pruzzo, Natalia Andrusko, Mónica Hourcade, Guillermo Labadie*. A&G, 81, (2010)
30- Parallel solution synthesis of lavendustin analogs as antileishmanial agents Diego G. Ghiano, Paulo B. Carvalho, Babu L. Tekwani, Mitchell A. Avery, Guillermo Labadie*. Arkivoc vii, 297-311 (2011).
31- An entry to curcuphenol/elvirol core structures via a retro-aldol procedure. María Fernanda Plano, Guillermo R. Labadie, Melissa R. Jacob, Babu L. Tekwani, and Raquel M. Cravero. Chem. Biodivers. 8, 1098-1111, (2011). doi: 10.1002/cbdv.201000160
32- Simplified tricycle model of quassinoids with in vitro antiparasitic activity. María F. Plano, Guillermo R. Labadie, Babu Tekwani, Raquel M. Cravero. Arkivoc vii, 477-489 (2011).
33- Targeting tuberculosis through a small focused library of 1,2,3-triazoles. Guillermo R. Labadie*, Agustina de la Iglesia, Héctor R. Morbidoni. Mol. Divers. 15, 1017-1024 (2011). doi: 10.1007/s11030-011-9319-0
34- Synthesis and antikinetoplastid activity of a series of N,N’-substituted diamines. Andrea P. Caminos, Esteban A. Panozzo-Zenere, Shane Wilkinson, Babu Tekwani, and Guillermo R. Labadie*. Bioorg. Med. Chem. Lett. 22, 1712-1715 (2012) doi: 10.1016/j.bmcl.2011.12.101
35- Synthesis and biological activity profile of novel 2-cinnamylidene-cycloalkane-1,3-diones related to coruscanone A: Promising new antileishmanial agents. Martín J. Riveira, Babu Tekwani, Guillermo R. Labadie,*and Mirta P. Mischne.* MedChemComm 3, 1294-1298 (2012) doi: 10.1039/C2MD20143G
36- Chemobiosynthesis of new antimalaric macrolides. Mariana Useglio, Christopher D. Goodman, Salvador Peirú, Guillermo R. Labadie, Geoffrey I. McFadden, Hugo Gramajo and Eduardo Rodríguez. Antimicrob. Agents Chemother. 57, 907-13. (2013) doi:10.1128/AAC.01825-12
37- Regioselective Covalent Immobilization of Catalytically Active Glutathione S-Transferase on Glass Slides. Rajesh Viswanathan, Guillermo R. Labadie, and C. Dale Poulter. Bioconjug. Chem..(2013) doi: 10.1021/bc300462j
38- Identification of a bifunctional C- and O-glucosyltransferase in maize. María Lorena Falcone-Ferreyra, Eduardo Rodriguez, María Isabel Casas, Guillermo Labadie, Erich Grotewold, and Paula Casati. J. Biol. Chem. 288, 31678-31688 (2013) doi: 10.1074/jbc.M113.510040
39- Click chemistry decoration of amino sterols as promising strategy to developed new leishmanicidal drugs. Exequiel O. J. Porta, Paulo Carvalho, Babu Tekwani, Mitchell A. Avery, and Guillermo R. Labadie.* Steroids 74, 28-36 (2014) doi: 10.1016/j.steroids.2013.10.010
40- Identification of Novel Chemical Scaffolds Inhibiting Trypanothione Synthetase from Pathogenic Trypanosomatids. Diego Benítez, Andrea Medeiros, Lucía Fiestas, Esteban A. Panozzo-Zenere, Franzisca Maiwald, Theodora Calogeropoulou, Anastasia Detsi, Marina Roussaki, Kyriakos C. Prousis, Timo Jaeger, Jonas Šarlauskas, Lucíja Peterlin Mašič, Conrad Kunick, Guillermo R. Labadie, Leopold Flohe, Marcelo A. Comini* Plos Neglected Tropical Diseases 10 (4), e0004617 (2016). doi: 10.1371/journal.pntd.0004617.
41- Simple method for high purity acylated steryl glucosides synthesis. Sebastián N. Jäger, Martin Mittelbach, Rodolfo Cabrera, Guillermo R. Labadie.* Eur. J. Lip. Sci. Tech. 118, 827–833 (2016) doi: 10.1002/ejlt.201500205
42- Tuning acid catalyzed ortho-phenol prenylation as a molecular diversity tool. Sebastián N. Jäger, Exequiel O. J. Porta, and Guillermo R. Labadie* Mol. Diver. 20, 407-419 (2016) doi: 10.1007/s11030-015-9644-9
43- Antitubercular activity of 1,2,3-triazolyl fatty acid derivatives.Diego G. Ghiano, Agustina de la Iglesia, Nina Liu, Peter J. Tonge, Héctor R. Morbidoni, and Guillermo R. Labadie* Eur. J. Med. Chem. 125, 842–852 (2017). doi: 10.1016/j.ejmech.2016.09.086
44- Antitrypanosomal activity of prenyl-1,2,3-triazoles. Exequiel O. J. Porta, Sebastián N. Jäger, Isabel Nocito, Galina Lepesheva, Esteban Serra, Babu L. Tekwani and Guillermo R. Labadie* MedChemComm (2017) doi: 10.1039/C7MD00008A
23- An efficient approach toward the synthesis of the A/B rings of Ouabain. María Fernanda Plano, Guillermo R. Labadie, Manuel Gonzalez Sierra and Raquel M. Cravero. Tetrahedron Lett. 47, 7447-7449 (2006) doi: 10.1016/j.tetlet.2006.08.047
24- A simple synthesis of a model of the tetracyclic bis-ketal lactone mainframe of saudin. Guillermo R. Labadie, Liliana E. Luna, Raquel M. Cravero, Manuel González-Sierra Helv. Chim. Acta 89, 2732-2737 (2006) doi: 10.1021/ja061131o
25- Design, synthesis and evaluation of omega-azido and alkynyl farnesyl diphosphate analogs as protein farnesyl transferase substrates. Guillermo R. Labadie, Rajesh Viswanathan and C. Dale Poulter. J. Org. Chem. 72, 9291- 9297 (2007) doi: 10.1021/jo7017747
26- Semisynthetic Studies on the Manzamine Alkaloids. Khalid A. El Sayed, Ashraf A. Khalil, Muhammad Yousaf, Guillermo Labadie, Gundluru M. Kumar, Scott G. Franzblau, Alejandro M. S. Mayer, Mitchell A. Avery, and Mark T. Hamann. J. Nat. Prod. 71, 300-308 (2008) doi: 10.1021/np0703702
27- Preparation of phenyl-butyraldehydes using a base-catalyzed aromatization of dienones. María Fernanda Plano, Guillermo R. Labadie, Raquel M. Cravero. Tetrahedron Lett. 49, 2872–2874 (2008) doi: 10.1016/j.tetlet.2008.03.038
28- Biosynthesis of TDP-L-megosamine: pathway elucidation and megalomicin A production in Escherichia coli. Mariana Useglio, Salvador Peirú, Eduardo Rodríguez, Guillermo R. Labadie, John R. Carney, and Hugo Gramajo Appl. Environ. Microbiol. 76, 3869-3077 (2010) doi: 10.1128/AEM.03083-09
29- Identificación, cuantificación y determinación de variabilidad en el tiempo de componentes insolubles de biodiesel de soja comerciales argentinos. Rodolfo Cabrera, Pablo Pruzzo, Natalia Andrusko, Mónica Hourcade, Guillermo Labadie*. A&G, 81, (2010)
30- Parallel solution synthesis of lavendustin analogs as antileishmanial agents Diego G. Ghiano, Paulo B. Carvalho, Babu L. Tekwani, Mitchell A. Avery, Guillermo Labadie*. Arkivoc vii, 297-311 (2011).
31- An entry to curcuphenol/elvirol core structures via a retro-aldol procedure. María Fernanda Plano, Guillermo R. Labadie, Melissa R. Jacob, Babu L. Tekwani, and Raquel M. Cravero. Chem. Biodivers. 8, 1098-1111, (2011). doi: 10.1002/cbdv.201000160
32- Simplified tricycle model of quassinoids with in vitro antiparasitic activity. María F. Plano, Guillermo R. Labadie, Babu Tekwani, Raquel M. Cravero. Arkivoc vii, 477-489 (2011).
33- Targeting tuberculosis through a small focused library of 1,2,3-triazoles. Guillermo R. Labadie*, Agustina de la Iglesia, Héctor R. Morbidoni. Mol. Divers. 15, 1017-1024 (2011). doi: 10.1007/s11030-011-9319-0
34- Synthesis and antikinetoplastid activity of a series of N,N’-substituted diamines. Andrea P. Caminos, Esteban A. Panozzo-Zenere, Shane Wilkinson, Babu Tekwani, and Guillermo R. Labadie*. Bioorg. Med. Chem. Lett. 22, 1712-1715 (2012) doi: 10.1016/j.bmcl.2011.12.101
35- Synthesis and biological activity profile of novel 2-cinnamylidene-cycloalkane-1,3-diones related to coruscanone A: Promising new antileishmanial agents. Martín J. Riveira, Babu Tekwani, Guillermo R. Labadie,*and Mirta P. Mischne.* MedChemComm 3, 1294-1298 (2012) doi: 10.1039/C2MD20143G
36- Chemobiosynthesis of new antimalaric macrolides. Mariana Useglio, Christopher D. Goodman, Salvador Peirú, Guillermo R. Labadie, Geoffrey I. McFadden, Hugo Gramajo and Eduardo Rodríguez. Antimicrob. Agents Chemother. 57, 907-13. (2013) doi:10.1128/AAC.01825-12
37- Regioselective Covalent Immobilization of Catalytically Active Glutathione S-Transferase on Glass Slides. Rajesh Viswanathan, Guillermo R. Labadie, and C. Dale Poulter. Bioconjug. Chem..(2013) doi: 10.1021/bc300462j
38- Identification of a bifunctional C- and O-glucosyltransferase in maize. María Lorena Falcone-Ferreyra, Eduardo Rodriguez, María Isabel Casas, Guillermo Labadie, Erich Grotewold, and Paula Casati. J. Biol. Chem. 288, 31678-31688 (2013) doi: 10.1074/jbc.M113.510040
39- Click chemistry decoration of amino sterols as promising strategy to developed new leishmanicidal drugs. Exequiel O. J. Porta, Paulo Carvalho, Babu Tekwani, Mitchell A. Avery, and Guillermo R. Labadie.* Steroids 74, 28-36 (2014) doi: 10.1016/j.steroids.2013.10.010
40- Identification of Novel Chemical Scaffolds Inhibiting Trypanothione Synthetase from Pathogenic Trypanosomatids. Diego Benítez, Andrea Medeiros, Lucía Fiestas, Esteban A. Panozzo-Zenere, Franzisca Maiwald, Theodora Calogeropoulou, Anastasia Detsi, Marina Roussaki, Kyriakos C. Prousis, Timo Jaeger, Jonas Šarlauskas, Lucíja Peterlin Mašič, Conrad Kunick, Guillermo R. Labadie, Leopold Flohe, Marcelo A. Comini* Plos Neglected Tropical Diseases 10 (4), e0004617 (2016). doi: 10.1371/journal.pntd.0004617.
41- Simple method for high purity acylated steryl glucosides synthesis. Sebastián N. Jäger, Martin Mittelbach, Rodolfo Cabrera, Guillermo R. Labadie.* Eur. J. Lip. Sci. Tech. 118, 827–833 (2016) doi: 10.1002/ejlt.201500205
42- Tuning acid catalyzed ortho-phenol prenylation as a molecular diversity tool. Sebastián N. Jäger, Exequiel O. J. Porta, and Guillermo R. Labadie* Mol. Diver. 20, 407-419 (2016) doi: 10.1007/s11030-015-9644-9
43- Antitubercular activity of 1,2,3-triazolyl fatty acid derivatives.Diego G. Ghiano, Agustina de la Iglesia, Nina Liu, Peter J. Tonge, Héctor R. Morbidoni, and Guillermo R. Labadie* Eur. J. Med. Chem. 125, 842–852 (2017). doi: 10.1016/j.ejmech.2016.09.086
44- Antitrypanosomal activity of prenyl-1,2,3-triazoles. Exequiel O. J. Porta, Sebastián N. Jäger, Isabel Nocito, Galina Lepesheva, Esteban Serra, Babu L. Tekwani and Guillermo R. Labadie* MedChemComm (2017) doi: 10.1039/C7MD00008A